產(chǎn)品屬性:
產(chǎn)品名稱 | Leelamine |
規(guī)格 | 5mg、10mg、25mg、50mg |
貨號(hào) | EY-01Y20677 |
Cas No.: 1446-61-3
別名: N/A
化學(xué)名: N/A
分子式: C20H31N
分子量: 285.5
溶解度: DMF: 30 mg/ml,DMSO: 30 mg/ml,Ethanol: 100 mg/ml,Ethanol:PBS (pH 7.2) (1:3): .25 mg/ml
儲(chǔ)存條件: Store at -20°C
General tips:For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition:Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
Leelamine is a diterpene molecule whose name derives from the Sanskrit word leela which means "play". It has weak affinity for the human central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 μM. Leelamine inhibits pyruvate dehydrogenase kinase (PDK) with an IC50 value of 9.5 μM. Derivatives of leelamine exhibit anti-inflammatory activity and show moderate inhibition of phospholipase A2 activity from a variety of sources.
特別提醒公司產(chǎn)品僅供科研使用