產(chǎn)品屬性:
產(chǎn)品名稱 | RS 127445 hydrochloride |
規(guī)格 | 10 mg、50 mg |
貨號 | EY-01Y18036 |
Cas No.: 199864-86-3
別名: N/A
化學名: N/A
分子式: C17H16FN3.HCl
分子量: 317.79
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
High affinity 5-HT2B receptor antagonist (pKi = 9.5). Displays 1000-fold selectivity for 5-HT2B with good bioavailability.Bonhaus et al (1999) RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist. Br.J.Pharmacol. 127 1075 PMID:10455251 |Callebert et al (2006) Evidence for a control of plasma serotonin levels by 5-Hydroxytryptamine2B receptors in mice. J.Pharmacol.Exp.Ther. 317 724 PMID:16461587
特別提醒公司產(chǎn)品僅供科研使用