產品屬性：
產品名稱 | Thioperamide (maleate) |
規(guī)格 | 1mg、5mg、10mg、25mg |
貨號 | EY-01Y18025 |
Cas No.: 148440-81-7
別名: N/A
化學名: N-cyclohexyl-4-(1H-imidazol-5-yl)-1-piperidinecarbothioamide, 2Z-butenedioate
分子式: C15H24N4S?C4H4O4
分子量: 408.5
溶解度: 10mg/mL in ethanol, 25mg/mL in DMSO, 30mg/mL in DMF
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Thioperamide (maleate) is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier. This compound binds to rat cerebral cortical cells in vitro with a pKi value of 8.4 and inhibits histamine binding in vivo with an ED50 value of 1 mg/kg.[1] At a dose of 5 mg/kg thioperamide (maleate) inhibits kindled seizures in rats by decreasing histamine and gamma-aminobutyric acid.[2]
特別提醒公司產品僅供科研使用
