產(chǎn)品屬性:
產(chǎn)品名稱 | Teneligliptin hydrobromide hydrate |
規(guī)格 | 10mg、50mg |
貨號(hào) | EY-01Y11510 |
Cas No.: 1572583-29-9
別名: N/A
化學(xué)名: N/A
分子式: C22H30N6OS
分子量: 426.58
溶解度: DMF: 30 mg/ml,DMSO: 30 mg/ml,Ethanol: 2 mg/ml,PBS (pH 7.2): 10 mg/ml
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
Teneligliptin hydrobromide hydrate is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM[1].[1]. Fukuda-Tsuru S, et al. A novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor, teneligliptin, improves postprandial hyperglycemia and dyslipidemia after single and repeated administrations. Eur J Pharmacol. 2012 Dec 5;696(1-3):194-202.
特別提醒公司產(chǎn)品僅供科研使用